Oseltamavir: Difference between revisions

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==General==
#REDIRECT[[Oseltamivir]]
*Type: Antiviral - neuraminidase inhibitor
*Dosage Forms: capsule (30, 45, 75mg), powder for PO susp (6mg/mL)
*Common Trade Names: Tamiflu
 
==Adult Dosing==
===[[Influenza]]===
75mg PO BID x5d
 
==Pediatric Dosing==
''5 day course''
*1-8 months: 3mg/kg PO BID
*9-23 months: 3.5mg/kg PO BID
*2-12 years:
**<15kg: 30mg PO BID
**16-23kg: 45mg PO BID
**24-40kg: 60mg PO BID
**>40kg: 75mg PO BID
 
==Special Populations==
*[[Drug Ratings in Pregnancy|Pregnancy Rating]]: Category C
*Lactation: Unknown; caution required
*Renal Dosing
**Adult
**Pediatric
*Hepatic Dosing
**Adult
**Pediatric
 
==Contraindications==
*Allergy to class/drug
 
==Adverse Reactions==
===Serious===
Rare <1%
 
Arrhythmia, delirium, hemorrhagic colitis, hepatitis, seizure, TEN, SJS, angioedema, unstable angina, pseudomembranous colitis
 
===Common===
Abdominal pain, insomnia, nausea, vomitting, vertigo, epistaxis, ear complaints, conjunctivitis.
 
==Pharmacology==
*Half-life: 1-3 hrs (oseltamivir); 6-10hrs oseltamivir carboxylate)
*Metabolism: hepatic
*Excretion: urine/stool
*Mechanism of Action: competitive inhibition of influenza virus neuraminidase enzyme, effectively halting viral release from infected cells and passing through mucus membranes.
 
==See Also==
 
 
==References==
<references/>
 
[[Category:Pharmacology]]

Latest revision as of 00:45, 23 September 2019

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